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Raw Tianeptine powder (66981-73-5)

(1 customer review)

Tianeptine powder is a nootropic and an antidepressant selective serotonin re-uptake enhancer (SSRE). It is generally in ……..


Status: In Mass Production
Unit: 25kg/Drum
Capacity: 1190kg/month

Description

Raw Tianeptine powder (66981-73-5) video

Raw Tianeptine powder (66981-73-5)

Raw Tianeptine powder is an antidepressant agent with a novel neurochemical profile.Raw Tianeptine powder does not appear to be associated with adverse cognitive, psychomotor, sleep, cardiovascular or bodyweight effects and has a low propensity for abuse. Raw Tianeptine powder has a comparatively favourable pharmacokinetic profile. It is not subject to first-pass hepatic metabolism, has high bioavailability and limited distribution, and is rapidly eliminated. While this offers advantages for Raw Tianeptine powder over the tricyclic antidepressant agents in terms of dose titration, treatment changes and potential drug interactions, its rapid elimination makes adherence to dosage schedules more important. Raw Tianeptine powder differs from most antidepressants in that it is not primarily metabolised by the hepatic cytochrome P450 system, indicating less likelihood of drug-drug interactions; this is of particular interest for elderly patients.

Raw Tianeptine powder (66981-73-5) Specifications

Product Name Raw Tianeptine powder
Chemical Name Raw Tianeptine powder; 66981-73-5; 72797-41-2; Raw Tianeptine powder Acid; Raw Tianeptine powder
Brand Name Yocon
Drug Class depressive episodes
CAS Number 66981-73-5
InChIKey JICJBGPOMZQUBB-UHFFFAOYSA-N
Molecular Formula C21H25ClN2O4S
Molecular Weight 436.951 g/mol
Monoisotopic Mass 436.122 g/mol
Melting Point  148
Boiling Point 609.2
Biological Half-Life No date available
Color White to off-white powder
Solubility  No date available
Storage Temperature  Refrigerator
Application It is a drug used for treating major depressive episodes (mild, moderate, or severe).

 

Raw Tianeptine powder (66981-73-5) Description

Tianeptine powder is a drug primarily used to improve the symptoms of major depressive disorder (MDD). It has also been used to help irritable bowel syndrome and asthma. Structurally, it is classified as a tricyclic antidepressant (TCA), however, it possesses different pharmacological properties than typical tricyclic antidepressants. Tianeptine was discovered and patented by the French society of Medical Research in the 1960s. It’s brand names include Stablon, Coaxil. Tatinol, Tianeurax, and Salymbra.

Tianeptine powder does not appear to be associated with adverse cognitive, psychomotor, sleep, cardiovascular or bodyweight effects and has a low propensity for abuse. Raw Tianeptine powder has a comparatively favourable pharmacokinetic profile. It is not subject to first-pass hepatic metabolism, has high bioavailability and limited distribution, and is rapidly eliminated. While this offers advantages for Raw Tianeptine powder over the tricyclic antidepressant agents in terms of dose titration, treatment changes and potential drug interactions, its rapid elimination makes adherence to dosage schedules more important. Raw Tianeptine powder differs from most antidepressants in that it is not primarily metabolised by the hepatic cytochrome P450 system, indicating less likelihood of drug-drug interactions; this is of particular interest for elderly patients.

Recently, Tianeptine is available in European, Asian, and South American countries. It is banned in the United Kingdom and is not medically prescribed by doctors in the United States.

Tianeptine powder (66981-73-5) Mechanism of Action

Recent studies suggest that tianeptine acts as a full agonist at the mu-type opioid receptor (MOR). The mu opioid receptors are currently being studied as effective targets for antidepressant therapies. It is believed that the clinical effects of tianeptine are owed to its modulation of these receptors. In addition to its actions on the opioid receptor, previous studies have owed its action to its effect on the serotonin receptor dopamine (D2/3) receptors and glutamate receptors.

Tianeptine powder is a unique antidepressant and anxiolytic medication that stimulates the uptake of serotonin (5-hydroxytryptamine; 5-HT), and 5-hydroxyindoleacetic acid (5-HIAA) in brain tissue.

Although the monoaminergic neurotransmitters serotonin (5-HT), noradrenaline (NA) and dopamine (DA) are proven to be related to the occurrence of depressive disorders, it is now recognized that monoamine deficits are not sufficient to explain the mechanism of action of antidepressant medications.

Application of Tianeptine powder (66981-73-5)

▪ Tianeptine improve the symptoms of major depressive disorder (MDD)

▪ Tianeptine help irritable bowel syndrome and asthma

▪ Tianeptine improve mood and soothes anxiety.

▪ Tianeptine increases how much serotonin the brain absorbs

▪ Tianeptine enhance motivation, focus and cognitive, suppress anxiety, rejuvenation and reduce cognitive fatigue.

Recommended Tianeptine powder (66981-73-5) Dosage

Tianeptine powder is generally prescribed at a dose of 12.5 mg and taken three times per day. Unlike other TCAs and selective serotonin reuptake inhibitors (SSRIs), tianeptine doses do not need to be increased slowly and a taper when the medication is discontinued is not required.

Side effects of Tianeptine powder (66981-73-5)

The side effects of tianeptine powder are surprisingly limited. Compared to other TCAs and even the SSRI class of antidepressants, tianeptine powder is almost free of side effects. Despite its mild side effect profile, it is important not to mix tianeptine with monoamine oxidase inhibitors or other antidepressants as the combinations could be life threatening. Tianeptine should also not be mixed with anesthetics and its use should cease 24-48 prior to surgical intervention requiring anesthetics or hypnotics. Here are a few of the more common side effects associated with tianeptine.

 Constipation

 Diarrhea

 Indigestion

 Vomiting

 Dry mouth

 Fatigue

 Insomnia

 Changes in appetite

 Dizziness

 Respiratory depression

 Sleepiness

 Blurred vision

 Decreased sex drive

 Headache

 Itching

 


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1 review for Raw Tianeptine powder (66981-73-5)

  1. phcoker

    Got Raw Tianeptine powder to test, test result show very high quality and purity!

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