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Endurobol (317318-70-0)

Endurobol is a PPARδ receptor. It activates the same pathways activated through exercise, including PPARδ and AMP……..


Status: In Mass Production
Unit: 25kg/Drum
Capacity: 1290kg/month

Description

Endurobol (317318-70-0) video

 

Endurobol (317318-70-0) Description

Endurobol is a PPARδ receptor. It activates the same pathways activated through exercise, including PPARδ and AMP-activated protein kinase. It had been investigated as a potential treatment for obesity, diabetes, dyslipidemia and cardiovascular disease. Endurobol has a synergistic effect when combined with AICAR: the combination has been shown to significantly increase exercise endurance in animal studies more than either compound alone.

Endurobol could be used by athletes as an ergogenic performance enhancing drug that was not currently controlled by regulations or detected by standard tests. One of the main researchers from the study on enhanced endurance consequently developed a urine test to detect the drug, and made it available to the International Olympic Committee.

Endurobol (317318-70-0) Specifications

Product Name Endurobol
Chemical Name 2-[2-methyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]acetic acid;GW-501615;CB6465728;2-(4-((2-(4-(Trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylthio)-2-methylphenoxy)acetic a;GW1516; GSK-516.
Brand Name Endurobol
Drug Class Inhibitors;Intermediates & Fine Chemicals; Pharmaceuticals;Sulfur & Selenium Compounds;kl; Inhibitor;Antineoplastic;SARMs(Selective androgen receptor modulator);Sarms
CAS Number 317318-70-0
InChIKey YDBLKRPLXZNVNB-UHFFFAOYSA-N
Molecular Formula C21H18F3NO3S2
Molecular Weight 453.494 g/mol
Monoisotopic Mass 453.068 g/mol
Melting Point 134-136°C
Boiling Point  584.543ºc at 760mmhg
Biological Half-Life 16-24 hours
Color white to beige
Solubility  DMSO: soluble20mg/mL, clear
Storage Temperature  Refrigerator
Endurobol Application A selective and potent PPARβ agonist;An experimental drug meant to control lipids and increase the level of HDL, or good cholesterol, in the bloodstream. A cell-permeable, thiazolyl compound that acts as a potent, high affinity, PPARδ agonist.

 


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